An Integrated in Silico 3D Model-Driven Discovery of a Novel, Potent, and Selective Amidosulfonamide 5-HT<sub>1A</sub> Agonist (PRX-00023) for the Treatment of Anxiety and Depression

Oren M. Becker(Epix Pharmaceuticals (United States)), Silvia Noiman(Epix Pharmaceuticals (United States)), Pradyumna Mohanty(Epix Pharmaceuticals (United States)), Dale Dhanoa(Epix Pharmaceuticals (United States)), Raphael Nudelman(Teva Pharmaceuticals (Israel)), Sharon Shacham(Roche (Switzerland)), Alexander Heifetz(Argonne National Laboratory), Anurag Sharadendu(Epix Pharmaceuticals (United States)), Srinivasa R. Cheruku(Epix Pharmaceuticals (United States)), Dongli Chen(Epix Pharmaceuticals (United States)), Yael Marantz(Epix Pharmaceuticals (United States)), Michael Kauffman(Roche (Switzerland)), Merav Fichman(Epix Pharmaceuticals (United States))
Journal of Medicinal Chemistry
May 9, 2006
Cited by 141


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