Identification of <i>N</i>,1,4,4-Tetramethyl-8-{[4-(4-methylpiperazin-1-yl)phenyl]amino}-4,5-dihydro-1<i>H</i>-pyrazolo[4,3-<i>h</i>]quinazoline-3-carboxamide (PHA-848125), a Potent, Orally Available Cyclin Dependent Kinase Inhibitor

Maria Gabriella Brasca(Nerviano Medical Sciences), Marina Ciomei(Nerviano Medical Sciences), Paolo Pevarello(Nerviano Medical Sciences), Walter Moretti(Nerviano Medical Sciences), Dario Ballinari(Nerviano Medical Sciences), Francesco Colotta(Humanitas University), Ciro Mercurio(Mylan (Switzerland)), Giovanni Cervi(Nerviano Medical Sciences), Valter Croci(Nerviano Medical Sciences), Francesca Quartieri(Nerviano Medical Sciences), Wilma Pastori(Nerviano Medical Sciences), Achille Panzeri(Nerviano Medical Sciences), Alexander D. Cameron(University of Warwick), Maristella Colombo(Nerviano Medical Sciences), Paola Vianello(Nerviano Medical Sciences), Roberto D’Alessio(Nerviano Medical Sciences), Elena Casale, Gabriella Traquandi(Nerviano Medical Sciences), Anna Vulpetti(Nerviano Medical Sciences), Fulvia Roletto(Nerviano Medical Sciences), Nadia Amboldi(University of Pavia), Francesco Fiorentini(Nerviano Medical Sciences), Antonella Isacchi(Nerviano Medical Sciences)
Journal of Medicinal Chemistry
July 15, 2009
Cited by 128


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