Discovery and optimization of Lu AF58801, a novel, selective and brain penetrant positive allosteric modulator of alpha-7 nicotinic acetylcholine receptors: Attenuation of subchronic phencyclidine (PCP)-induced cognitive deficits in rats following oral administration
Jørgen Eskildsen(Lundbeck (Denmark)), Jesper F. Bastlund(Lundbeck (Denmark)), M.L. Laursen(Lundbeck (Denmark)), Roger L. Papke(Io Therapeutics (United States)), Jette Bisgaard Boll(Lundbeck (Denmark)), John P. Redrobe(Douglas Mental Health University Institute), Anette Sams(Glostrup Hospital), Kim Dekermendjian(Lundbeck (Denmark)), Kristen Frederiksen(Mayo Clinic in Florida), Christoffer Bundgaard(University of North Carolina at Chapel Hill)
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