Malonate-based inhibitors of mammalian serine racemase: Kinetic characterization and structure-based computational study

Barbora Vorlová(Charles University), Martin Lepšı́k(Centre National de la Recherche Scientifique), Pavel Hobza(Czech Academy of Sciences, Institute of Organic Chemistry and Biochemistry), Petr Jansa(Czech Academy of Sciences, Institute of Organic Chemistry and Biochemistry), Michal Otyepka(VSB - Technical University of Ostrava), Jan Konvalinka(Institute of Organic Chemistry), Jana Jirásková-Vaníčková(Charles University), Jan Řezáč(Czech Academy of Sciences), Dana Nachtigallová(University of Vienna), Jindřich Fanfrlík(Czech Academy of Sciences), Haresh Ajani(Regional Centre of Advanced Technologies and Materials)
European Journal of Medicinal Chemistry
October 16, 2014
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