Phospshoinositide 3-Kinase (PI3K)/Mammalian Target of Rapamycin (mTOR) Dual Inhibitors: Discovery and Structure–Activity Relationships of a Series of Quinoline and Quinoxaline Derivatives

Nobuko Nishimura(Amgen (United States)), Mark H. Norman(Amgen (United States)), Raju Subramanian(Gilead Sciences (United States)), Nancy R. Zhang(University of the Arts), Kevin Yang(Revolution Medicines (United States)), Leeanne Zalameda(Amgen (United States)), Tisha San Miguel(Amgen (United States)), Douglas A. Whittington(Amgen (United States)), Erin L. Mullady(Amgen (United States)), Marian C. Bryan(Johnson & Johnson (United States)), Shon K. Booker(Amgen (United States)), Longbin Liu(National University of Defense Technology), Ling Wang(Amgen (United States)), Hongyu Liao, Paul E. Hughes(Amgen (United States)), Sean Caenepeel(Amgen (United States)), Kristin L. Andrews(Amgen (United States)), Aaron Siegmund(Amgen (United States)), Yunxin Bo(Amgen (United States)), John D. McCarter(Amgen (United States)), Daniel J. Freeman(Amgen (United States)), Nuria Tamayo(Amgen (United States))
Journal of Medicinal Chemistry
May 25, 2011
Cited by 60


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