Evaluation of a Series of Naphthamides as Potent, Orally Active Vascular Endothelial Growth Factor Receptor-2 Tyrosine Kinase Inhibitors
Matthew M. Weiss(Amgen (United States)), Roger Zanon(Amgen (United States)), David Bauer(Amgen (United States)), Michael Schrag(Amgen (United States)), Danlin Chen(Amgen (United States)), Julie Flynn(Amgen (United States)), Juan Estrada(Amgen (United States)), Douglas A. Whittington(Amgen (United States)), George Borg(Aalborg University), Andrew S. Tasker(Amgen (United States)), Jean-Christophe Harmange(Amgen (United States)), Anthony Polverino(Amgen (United States)), Deborah M. Choquette(Amgen (United States)), Tom DeMelfi(Amgen (United States)), Charlie Starnes(Amgen (United States)), Michele Potashman(Biogen (United States)), Russell F. Graceffa(Amgen (United States)), Phillip M. Roveto(Amgen (United States)), Shawn Harriman(Amgen (United States)), James Bready(Amgen (United States)), Alexander Long(Amgen (United States)), Vinod F. Patel(Guy's Hospital), Daniel S. La(Amgen (United States)), Nicholas Doerr(Amgen (United States)), Virginia Berry(Amgen (United States)), Kelly Regal(Amgen (United States)), Loren Berry(Amgen (United States)), Yohannes Teffera(Amgen (United States)), Angela Coxon(Amgen (United States)), Stephen A. Kaufman(Amgen (United States)), Sesha Neervannan(Amgen (United States))
Cited by 34
Related Papers
Remarkably Stable Tetrahedral Intermediates: Carbinols from Nucleophilic Additions to<i>N</i>���Acylpyrroles
|Angewandte Chemie International Edition|2002|167
Apo2L/TRAIL and the Death Receptor 5 Agonist Antibody AMG 655 Cooperate to Promote Receptor Clustering and Antitumor Activity
|Cancer Cell|2014|155
One-pot asymmetric synthesis of tert-butanesulfinyl-protected amines from ketones by the in situ reduction of tert-butanesulfinyl ketimines
|Tetrahedron Letters|1999|111
Health-related quality of life in people with predementia Alzheimer’s disease, mild cognitive impairment or dementia measured with preference-based instruments: a systematic literature review
|Alzheimer s Research & Therapy|2020|104
Asymmetric synthesis of pre-protected α,α-disubstituted amino acids from tert-butanesulfinyl ketimines
|Tetrahedron Letters|2001|77