Design, synthesis, and structure–activity relationships of piperidine and dehydropiperidine carboxylic acids as novel, potent dual PPARα/γ agonists
Xiang‐Yang Ye(Hangzhou Normal University), Peter T. W. Cheng(Bristol-Myers Squibb (United States)), Jonathan Lippy(Bristol-Myers Squibb (United States)), Denis E. Ryono(Institut des Maladies Métaboliques et Cardiovasculaires), Narayanan Hariharan(Bristol-Myers Squibb (United States)), Celeste Twamley(Bristol-Myers Squibb (United States)), Robert Zahler(Institut des Maladies Métaboliques et Cardiovasculaires), Li‐Qun Gu(Texas A&M Health Science Center), Kenneth T. Locke(Medicines Evaluation Unit), Yixin Li(Baylor College of Medicine), Litao Zhang(Tianjin University of Traditional Chinese Medicine), Neil Flynn(Bristol-Myers Squibb (United States)), Kevin O’Malley(Medicines Evaluation Unit), Dennis Farrelly(Bristol-Myers Squibb (United States))
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