Catalytic in vivo protein knockdown by small-molecule PROTACs

Daniel P. Bondeson(Yale University), Alina Mares(Age UK), Ian E. Smith(Age UK), Eunhwa Ko(Yale University), Sébastien Campos(Age UK), Afjal H. Miah(Age UK), Katie E Mulholland(Age UK), Natasha Routly(Age UK), Dennis L. Buckley(Yale University), Jeffrey L. Gustafson(Yale University), Nico Zinn, Paola Grandi, Satoko Shimamura, Giovanna Bergamini, Maria Faelth-Savitski, Marcus Bantscheff, Carly S. Cox(Yale University), Deborah A. Gordon(Arvinas (United States)), Ryan R. Willard(Arvinas (United States)), John J. Flanagan(Arvinas (United States)), Linda Casillas(GlaxoSmithKline (United States)), Bartholomew J. Votta(GlaxoSmithKline (United States)), Willem den Besten(California Institute of Technology), Kristoffer Famm(Age UK), Laurens Kruidenier(Age UK), Paul S. Carter(Age UK), John D. Harling(Age UK), Ian Churcher(Age UK), Craig M. Crews(Yale University)
Nature Chemical Biology
June 10, 2015
Cited by 1,294Open Access
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