Discovery of N-(4-aryl-5-aryloxy-thiazol-2-yl)-amides as potent RORγt inverse agonists

Yonghui Wang(Weifang People's Hospital), Xichen Lin(GlaxoSmithKline (China)), Ling Zhou(GlaxoSmithKline (China)), Yingli Ma(GlaxoSmithKline (China)), Qianqian Wu(GlaxoSmithKline (China)), Ziqiang Cheng(Shandong Agricultural University), Qian Liu(Guangxi Medical University), Yi Li(Baylor College of Medicine), Wei Zhang(Capital Medical University), Lisa A. Orband‐Miller(GlaxoSmithKline (China)), Ting Yang(GlaxoSmithKline (China)), Liuqing Yang(GlaxoSmithKline (China)), Feng Ren(Henan Medical University), John D. Elliott(GlaxoSmithKline (China)), Stewart Leung(GlaxoSmithKline (China)), Zhijun Xiang(GlaxoSmithKline (China)), Sijie Lu(GlaxoSmithKline (China)), Jia‐Ning Xiang(GlaxoSmithKline (China)), Kathleen Zhang(GlaxoSmithKline (China))
Bioorganic & Medicinal Chemistry
August 1, 2015
Cited by 32


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