3-Aminopyrrolidinone Farnesyltransferase Inhibitors: Design of Macrocyclic Compounds with Improved Pharmacokinetics and Excellent Cell PotencyIan M. Bell, C. Blair Zartman, W. Wayt Gibbs et al.|Journal of Medicinal Chemistry|2002Cited by 86
Dual Protein Farnesyltransferase−Geranylgeranyltransferase-I Inhibitors as Potential Cancer Chemotherapeutic AgentsS. J. DESOLMS, Jeffrey S. Taylor, Terrence M. Ciccarone et al.|Journal of Medicinal Chemistry|2003Cited by 60
An allosteric Akt inhibitor effectively blocks Akt signaling and tumor growth with only transient effects on glucose and insulin levels in vivoCraig Cherrin, Hans E. Huber, Kathleen Haskell et al.|Cancer Biology & Therapy|2010Cited by 59
Potent inhibitors of farnesyltransferase and geranylgeranyltransferase-IDiem N. Nguyen, Carolyn A. Buser, Craig A. Stump et al.|Bioorganic & Medicinal Chemistry Letters|2002Cited by 22
2-Arylindole-3-acetamidesB. Wesley Trotter, Christopher J. Dinsmore, Amy G. Quigley et al.|Bioorganic & Medicinal Chemistry Letters|2001Cited by 19