Discovery of Imidazo[1,2-<i>b</i>]pyridazine Derivatives: Selective and Orally Available Mps1 (TTK) Kinase Inhibitors Exhibiting Remarkable Antiproliferative ActivityKen‐ichi Kusakabe, Yusuke Nakamura, Genta Tadano et al.|Journal of Medicinal Chemistry|2015Cited by 64
Indazole-Based Potent and Cell-Active Mps1 Kinase Inhibitors: Rational Design from Pan-Kinase Inhibitor Anthrapyrazolone (SP600125)Ken‐ichi Kusakabe, Yusuke Nakamura, Nobuyuki Ide et al.|Journal of Medicinal Chemistry|2013Cited by 47
Diaminopyridine-Based Potent and Selective Mps1 Kinase Inhibitors Binding to an Unusual Flipped-Peptide ConformationKen‐ichi Kusakabe, Yusuke Nakamura, Nobuyuki Ide et al.|ACS Medicinal Chemistry Letters|2012Cited by 33
A unique hinge binder of extremely selective aminopyridine-based Mps1 (TTK) kinase inhibitors with cellular activityKen‐ichi Kusakabe, Yusuke Nakamura, Nobuyuki Ide et al.|Bioorganic & Medicinal Chemistry|2015Cited by 20