Sequential Metabolism of AMG 487, a Novel CXCR3 Antagonist, Results in Formation of Quinone Reactive Metabolites That Covalently Modify CYP3A4 Cys239 and Cause Time-Dependent Inhibition of the EnzymeKirk R. Henne, Bradley K. Wong, Brooke M. VandenBrink et al.|Drug Metabolism and Disposition|2012Cited by 42