Discovery and Characterization of 6-{4-[3-(<i>R</i>)-2-Methylpyrrolidin-1-yl)propoxy]phenyl}-2<i>H</i>-pyridazin-3-one (CEP-26401, Irdabisant): A Potent, Selective Histamine H<sub>3</sub>Receptor Inverse AgonistRobert L. Hudkins, Michael Williams, Ming Tao et al.|Journal of Medicinal Chemistry|2011Cited by 68
CEP-26401 (Irdabisant), a Potent and Selective Histamine H3 Receptor Antagonist/Inverse Agonist with Cognition-Enhancing and Wake-Promoting ActivitiesRita Raddatz, Michael Williams, Siyuan Le et al.|Journal of Pharmacology and Experimental Therapeutics|2011Cited by 58
Synthesis and Biological Profile of the pan-Vascular Endothelial Growth Factor Receptor/Tyrosine Kinase with Immunoglobulin and Epidermal Growth Factor-Like Homology Domains 2 (VEGF-R/TIE-2) Inhibitor 11-(2-Methylpropyl)-12,13-dihydro-2-methyl-8-(pyrimidin-2-ylamino)-4<i>H</i>-indazolo[5,4-a]pyrrolo[3,4-c]carbazol-4-one (CEP-11981): A Novel Oncology Therapeutic AgentRobert L. Hudkins, Bruce Ruggeri, Mark A. Ator et al.|Journal of Medicinal Chemistry|2011Cited by 42