MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 7: Highly soluble and in vivo active quaternary ammonium analogue D13-9001, a potential preclinical candidateKen‐ichi Yoshida, William J. Watkins, Hironobu Nitanai et al.|Bioorganic & Medicinal Chemistry|2007Cited by 130
An ultrasensitive biosensor for high-resolution kinase activity imaging in awake miceJinfan Zhang, Bian Liu, Ingie Hong et al.|Nature Chemical Biology|2020Cited by 110
MexAB-OprM-Specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 1: Discovery and early strategies for lead optimizationKiyoshi Nakayama, William J. Watkins, Yohei Ishida et al.|Bioorganic & Medicinal Chemistry Letters|2003Cited by 82
MexAB-OprM specific efflux pump inhibitors in Pseudomonas aeruginosa. Part 3: Optimization of potency in the pyridopyrimidine series through the application of a pharmacophore modelKiyoshi Nakayama, William J. Watkins, Haruko C. Kawato et al.|Bioorganic & Medicinal Chemistry Letters|2003Cited by 65
Diffusing protein binders to intrinsically disordered proteinsCaixuan Liu, David Baker, Kejia Wu et al.|Nature|2025Cited by 42